Alpha-adrenergic agonist. Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has two subclasses 1 and 2. Alpha 2 receptors are associated with sympatholytic properties. Alpha-adrenergic agonists have the opposite function of alpha blockers.
Alpha-nists or alpha-2 adrenoceptor agonists are drugs used to treat high blood pressure. Centrally acting alpha-nists stimulate alpha
Drug class listed Drug name in publication Actual drug class Apraclonidine Adrenergic agonist [Alpha.sub.2]-agonist Brimonidine (ophthalmic) Adrenergic agonist [Alpha.sub.2]-agonist; antiglaucoma Dapiprazole Miotic Alpha-blocker Dipivefrine Prostaglandin Prodrug of epinephrine Naphazoline (ophthalmic) Decongestant [Alpha.sub.1]-agonist
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Alpha agonists are drugs that activate alpha adrenergic receptors . 2. type. 2.1. alpha nist. Alpha 1 receptors contract vascular smooth
Alpha agonists that stimulate alpha-2 receptors in the eye are effective at reducing intraocular pressure and glaucoma. Examples of alpha-2 adrenergic agonists: Brimonidine. Clonidine. Dexmedetomidine. Guanfacine. Methyldopa. Naphazoline. Lofexidine. Tizanidine. Nonspecific alpha adrenergic receptor agonists
List of references. Aantaa, Molecular pharmacology of alpha 2 alpha(2)-adrenoceptor agonist with local mode of action, Eur. J. Pharmacol
Adrenergic Agonists ; Tizanidine, An alpha-2 adrenergic agonist used for the short-term treatment of muscle spasticity. ; Methoxamine, An alpha adrenergic agonist
Alpha-agonists used therapeutically are relatively selective or non-selective for 1 or 2-adrenoceptors.Besides the drugs listed below, there are sympathomimetic drugs that have -agonist and -adrenoceptor agonist properties.
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